他莫西芬,99% CAS號:10540-29-1 廠家現(xiàn)貨供應-廣東大小化工-日韓一卡二卡三卡四卡免費觀在線_國產(chǎn)免費久久久精品
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- 廣東大小化工有限公司
Tamoxifen is a selective estrogen response modifier (SERM), proteinkinase C inhibitor and anti-angiogenetic factor. Tamoxifen is aprodrug that is metabolized to active metabolites4-hydroxytamoxifen (4-OHT) and endoxifen by cytochrome P450isoforms CYP2D6 and CYP3A4. In breast cancer, the gene repressoractivity of tamoxifen against ERBB2 is dependent upon PAX2. Blocksestradiol-stimulated VEGF production in breast tumorcells.\nProtein kinase C inhibitor. Induces apoptosis in humanmalignant glioma cell lines. Tamoxifen and its metabolite4-hydroxytamoxifen are selective estrogen response modifiers(SERMs) that act as estrogen antagonists in mammary gland. Blocksestradiol-stimulated VEGF production in breast tumorcells.
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